Iodo-Cycloisomerization of Aryl(indol-3-yl)methane-Tethered Propargyl Alcohols to 3-Iodocarbazoles via Selective 1,2-Alkyl Migration

dc.contributor.author Yaragorla, Srinivasarao
dc.contributor.author Bag, Debojyoti
dc.contributor.author Dada, Ravikrishna
dc.contributor.author Jose, K. V.Jovan
dc.date.accessioned 2022-03-27T08:49:27Z
dc.date.available 2022-03-27T08:49:27Z
dc.date.issued 2018-11-07
dc.description.abstract Herein, we disclose the first report on iodo-cycloisomerization of 1-(indol-3-yl)-1-arylbut-3-yn-2-ols to form 3-iodocarbazoles. The synthesis proceeds through a cascade 5-endo-spirocyclization, followed by selective 1,2-alkyl migration. This method governs the green synthesis principles such as open-flask reaction, AcOEt as the solvent, rt reaction with short time, use of iodine, and broad substrate scope with atom and step economy.
dc.identifier.citation ACS Omega. v.3(11)
dc.identifier.uri 10.1021/acsomega.8b02393
dc.identifier.uri https://pubs.acs.org/doi/10.1021/acsomega.8b02393
dc.identifier.uri https://dspace.uohyd.ac.in/handle/1/11874
dc.title Iodo-Cycloisomerization of Aryl(indol-3-yl)methane-Tethered Propargyl Alcohols to 3-Iodocarbazoles via Selective 1,2-Alkyl Migration
dc.type Journal. Article
dspace.entity.type
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